Efficacy and safety of maintenance therapy with pamiparib versus placebo for advanced gastric cancer responding to first-line platinum-based chemotherapy: Phase 2 study results


Por: Ciardiello F, Bang Y, Cervantes A, Dvorkin M, Lopez C, Metges J, Ruiz A, Calvo M, Strickland A, Kannourakis G, Muro K, Kawakami H, Wei J, Borg C, Zhu Z, Gupta N, Pelham R, Shen L

Publicada: 1 jun 2023 Ahead of Print: 1 jun 2023
Resumen:
BackgroundPoly (ADP-ribose) polymerase (PARP) inhibitors (PARPi) are approved for the treatment of various solid tumors. In gastric cancer, genes commonly harbor mutations in the homologous recombination DNA repair pathway, potentially increasing sensitivity to PARPi. Pamiparib (BGB-290) is a small molecule inhibitor of PARP1 and PARP2.MethodsThe PARALLEL-303 study (NCT03427814) investigated the efficacy and safety of pamiparib 60 mg orally (PO) twice daily (BID) versus placebo PO BID as maintenance therapy in patients with inoperable locally advanced or metastatic gastric cancer that responded to platinum-based first-line chemotherapy. The primary endpoint of this double-blind, randomized, global phase 2 study was progression-free survival (PFS) (RECIST version 1.1; per investigator assessment). Secondary endpoints included overall survival (OS) and safety.ResultsIn total, 136 patients were randomized 1:1 to receive pamiparib (n = 71) or placebo (n = 65). Median PFS was numerically longer with pamiparib versus placebo but did not reach statistical significance (3.7 months [95% confidence interval (CI): 1.9, 5.3] vs. 2.1 months [95% CI: 1.9, 3.8]; hazard ratio 0.8 [95% CI: 0.5, 1.2]; p = 0.1428). Median OS was 10.2 months (95% CI: 8.7, 16.3) in the pamiparib arm versus 12.0 months (95% CI: 8.2, not estimable) in the placebo arm. Overall, 8 patients (11.3%) in the pamiparib arm and 2 patients (3.1%) in the placebo arm experienced = 1 TEAE leading to treatment discontinuation.ConclusionsMaintenance pamiparib did not meet statistical significance for superiority versus placebo for PFS, but was well tolerated with few treatment discontinuations; no unexpected safety signals were identified.

Filiaciones:
Ciardiello F:
 Univ Campania Luigi Vanvitelli, Dipartimento Med Precis, Caserta, Italy

Bang Y:
 Seoul Natl Univ, Dept Internal Med, Coll Med, Seoul, South Korea

Cervantes A:
 Univ Valencia, Biomed Res Inst INCLIVA, Dept Med Oncol, CIBERONC, Valencia, Spain

Dvorkin M:
 St Petersburg Acad Univ, Russian Acad Sci, Algorithm Biol Lab, St Petersburg, Russia

Lopez C:
 Oregon Hlth & Sci Univ, Knight Canc Inst, Dept Med, Portland, OR USA

Metges J:
 CHU Morvan, Arpego Network, Inst Oncol & Haematol, Brest, France

Ruiz A:
 Hosp Puerta Hierro Majadohonda, Madrid, Spain

Calvo M:
 Inst Catala Oncol Hosp, Dept Med Oncol, ONCOBELL Program IDIBELL, Barcelona, Spain

Strickland A:
 Monash Univ, Dept Med Oncol, Monash Hlth, Melbourne, Vic, Australia

Kannourakis G:
 Ballarat Oncol & Haematol Serv, Wendouree, Vic, Australia

 Fiona Elsey Canc Res Inst, Ballarat, Vic, Australia

Muro K:
 Aichi Canc Ctr Hosp, Dept Clin Oncol, Nagoya, Japan

Kawakami H:
 Kindai Univ, Dept Med Oncol, Fac Med, Osaka, Japan

Wei J:
 Nanjing Univ, Comprehens Canc Ctr Drum Tower Hosp, Med Sch, Nanjing, Peoples R China

 Nanjing Univ, Clin Canc Inst, Nanjing, Peoples R China

Borg C:
 Univ Hosp Besancon, Med Oncol Dept, CIC BT1431, Besancon, France

 INSERM, Mol & Cellular Immune Therapies Canc, UMR1098, Besancon, France

Zhu Z:
 BeiGene Ltd, Clin Dev, Cambridge, MA USA

Gupta N:
 BeiGene Ltd, Clin Dev, Cambridge, MA USA

Pelham R:
 BeiGene Ltd, Clin Dev, Cambridge, MA USA

Shen L:
 Peking Univ Canc Hosp & Inst, Minist Educ Beijing, Dept Gastrointestinal Oncol, Key Lab Carcinogenesis & Translat Res, Beijing, Peoples R China

 Peking Univ Canc Hosp & Inst, Dept Gastrointestinal Oncol, 52 Fucheng Rd, Beijing 100142, Peoples R China
ISSN: 20457634





Cancer Medicine
Editorial
John Wiley and Sons Ltd, United States, Estados Unidos America
Tipo de documento: Article
Volumen: 12 Número: 12
Páginas: 13145-13154
WOS Id: 001000282300001
ID de PubMed: 37260158
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